4ksp A 2.93 BS01 1SU A 1 V470 A480 K482 E500 L504 I526 T528 W530 C531 G533 H573 F582 D593 F594 V24 A34 K36 E54 L58 I80 T82 W84 C85 G87 H127 F136 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S151 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=8.80, Kd=1.6nM IC50=77nM P15056 23906342 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLP 4ksp B 2.93 BS01 1SU B 1 V470 A480 K482 E500 L504 I526 T528 W530 C531 H573 F582 D593 F594 V24 A34 K36 E54 L58 I80 T82 W84 C85 H127 F136 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S152 2.7.11.1 0004672,0005524,0006468 IC50=77nM P15056 23906342 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 6oc1 A 2.7 BS03 1SU A 1 Y37 M42 Q46 H55 A58 F61 L66 L67 P68 Y355 L358 T359 P363 Y7 M12 Q16 H25 A28 F31 L36 L37 P38 Y325 L328 T329 P333 N144 F148 S214 N216 T217 K254 N283 N114 F118 S184 N186 T187 K224 N253 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 Q02127 31734178 404 TGDERFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLPRARFQDSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSPNTAGLRSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADH