4kkh A 2.0 BS01 1RQ A 1 I70 V78 A91 K93 I124 L144 M146 M149 N152 I26 V34 A47 K49 I80 L100 M102 M105 N108 D189 K191 N194 D207 T226 D145 K147 N150 D163 T180 2.7.11.24 0004672,0004707,0005524,0006468 Kd=46nM, IC50=1090nM P53779 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQKQLDEREHTIEEWKELIYKEVMN