4kbk A 2.1 BS01 1QG A 1 I15 I23 A36 K38 M80 M82 L85 G86 L135 I148 I13 I19 A32 K34 M70 M72 L75 G76 L125 I138 D128 K130 D118 K120 2.7.11.1,2.7.11.26 0004672,0005524,0006468 -logKd/Ki=8.18, IC50=6.6nM IC50=6.6nM P48730 23919824 401 LRVGNRYRLGRKIGSGGDIYLGTDIAAGEEVAIKLECQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 4kbk B 2.1 BS01 1QG B 1 I23 A36 K38 M80 M82 L85 G86 L135 I148 I21 A34 K36 M78 M80 L83 G84 L133 I146 D128 K130 D126 K128 2.7.11.1,2.7.11.26 0004672,0005524,0006468 IC50=6.6nM P48730 23919824 401 LRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 4kbk C 2.1 BS01 1QG C 1 I15 I23 A36 K38 M80 M82 L85 G86 L135 I148 I12 I17 A30 K32 M74 M76 L79 G80 L129 I142 D128 K130 D122 K124 2.7.11.1,2.7.11.26 0004672,0005524,0006468 IC50=6.6nM P48730 23919824 401 RVGNRYRLGRKIGSGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 4kbk D 2.1 BS01 1QG D 1 I15 I23 A36 K38 M80 M82 L85 G86 L135 I148 I13 I16 A29 K31 M68 M70 L73 G74 L123 I136 D128 K130 D116 K118 2.7.11.1,2.7.11.26 0004672,0005524,0006468 IC50=6.6nM P48730 23919824 401 LRVGNRYRLGRKIGDIYLGTDIAAGEEVAIKLECPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML