4k18 A 2.051 BS01 1OB A 1 G45 F49 V52 A65 K67 R122 L174 I185 D186 G14 F18 V21 A34 K36 R91 L143 I154 D155 D167 K169 N172 D186 L193 T204 D136 K138 N141 D155 L162 T173 2.7.11.1 0004672,0004674,0005524,0006468,0043066 Ki=1.1nM -logKd/Ki=8.96, Ki=1.1nM P11309 23623490 402 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLS