4k4j A 2.0 BS02 1O8 A 1 I268 A271 A272 Q275 F313 R316 L326 A327 I345 C432 L436 I24 A27 A28 Q31 F69 R72 L82 A83 I101 C188 L192 ? 0003677,0003707,0005634,0006355,0008270 -logKd/Ki=6.12, Kd=0.752uM EC50=820nM, Kd=33nM P19793 24187139 500 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP