4jlk A 1.89 BS02 1NO A 1 E53 V55 P89 F96 Q97 D133 F137 L141 S144 Y204 E34 V36 P60 F67 Q68 D104 F108 L112 S115 Y173 E53 R128 E34 R99 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0016310,0019136,0042803,0043771,0106383,1901135,1901293 IC50=18nM, Ki=9.5nM P27707 23947754 402 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4jlk A 1.89 BS03 1NO A 2 L82 Y86 R194 E196 E197 G199 I200 P201 Y204 L53 Y57 R163 E165 E166 G168 I169 P170 Y173 E53 R128 E34 R99 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0016310,0019136,0042803,0043771,0106383,1901135,1901293 IC50=18nM, Ki=9.5nM P27707 23947754 403 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4jlk B 1.89 BS02 1NO B 1 E53 V55 Y86 F96 Q97 D133 F137 Y204 E35 V37 Y59 F69 Q70 D106 F110 Y177 E53 R128 E35 R101 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0016310,0019136,0042803,0043771,0106383,1901135,1901293 IC50=18nM, Ki=9.5nM P27707 23947754 402 TRIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNVLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4jlk B 1.89 BS03 1NO B 2 S59 L82 Y86 E197 I200 P201 Y204 S41 L55 Y59 E170 I173 P174 Y177 E53 R128 E35 R101 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0016310,0019136,0042803,0043771,0106383,1901135,1901293 IC50=18nM, Ki=9.5nM P27707 23947754 403 TRIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNVLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL