2og8 A 2.3 BS01 1N8 A 1 A271 K273 E288 M292 L300 T316 Y318 M319 L371 A381 D382 F383 A35 K37 E52 M56 L64 T80 Y82 M83 L135 A145 D146 F147 D364 R366 A368 N369 D382 D128 R130 A132 N133 D146 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.5nM -logKd/Ki=9.30, IC50=0.5nM IC50=0.500000nM P06239 16970394 501 EWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFT 2og8 B 2.3 BS01 1N8 B 1 A271 E288 L300 T316 Y318 M319 Y360 L371 A381 D382 F383 A36 E53 L65 T81 Y83 M84 Y125 L136 A146 D147 F148 D364 R366 A368 N369 D382 D129 R131 A133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.5nM IC50=0.500000nM P06239 16970394 502 DEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLAPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTA