3ce3 A 2.4 BS01 1FN A 1 I1084 A1108 K1110 M1131 L1157 M1160 M1211 V1220 A1221 D1222 F1223 I31 A55 K57 M78 L104 M107 M158 V167 A168 D169 F170 D1204 A1206 R1208 N1209 D1222 A1243 D151 A153 R155 N156 D169 A176 2.7.10.1 0004672,0004713,0005524,0006468 ic50=1.8nM -logKd/Ki=8.74, IC50=1.8nM IC50=1.8nM P08581 18690676 1401 DLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 6oko A 2.1 BS01 1FN A 1 V36 A49 K51 E61 M65 F97 M98 L150 A160 D161 F162 V23 A36 K38 E48 M52 F84 M85 L137 A147 D148 F149 D143 K145 S147 N148 D161 T187 D130 K132 S134 N135 D148 T151 2.7.11.1 0004672,0005524,0006468 Q9QZL0 32184955 4000 VPLVSREELKKLEFVGKGGFGVVFRAHHRTWNHDVAVKIVNSKKISWEVKAMVNLRNENVLLLLGVTEDLQWDFVSGQALVTRFMENGSLAGLLQPEAPRPWPLLCRLLQEVVLGMCYLHSLDPPLLHRDLKPSNILLDPELHAKLADFGTLAYLDPELLFKVNLKASKASDVYSFGILVWAVLAGREAELVDQSRPPLTELPPGSPETPGLEKLKELMIHCWGSQSENRPSFQDCEPKTNEVYNLVKDKVDAAVSEVKHYLS 6oko B 2.1 BS01 1FN B 1 V36 A49 K51 E61 M65 L68 T95 F97 M98 L150 A160 D161 F162 V24 A37 K39 E49 M53 L56 T83 F85 M86 L138 A148 D149 F150 D143 K145 S147 N148 D161 D131 K133 S135 N136 D149 2.7.11.1 0004672,0005524,0006468 Q9QZL0 32184955 4000 AVPLVSREELKKLEFVGKGGFGVVFRAHHRTWNHDVAVKIVNSKKISWEVKAMVNLRNENVLLLLGVTEDLQWDFVSGQALVTRFMENGSLAGLLQPEAPRPWPLLCRLLQEVVLGMCYLHSLDPPLLHRDLKPSNILLDPELHAKLADFLAYLDPELLFKVNLKASKASDVYSFGILVWAVLAGREAELRQSRPPLTELPPGSPETPGLEKLKELMIHCWGSQSENRPSFQDCEPKTNEVYNLVKDKVDAAVSEVKHYLS