4i9i A 2.4 BS02 1DY A 1 H1184 G1185 F1188 A1191 G1196 D1198 H1201 Y1203 I1212 Y1213 F1214 A1215 S1221 Y1224 E1291 H81 G82 F85 A88 G93 D95 H98 Y100 I109 Y110 F111 A112 S118 Y121 E188 2.4.2.-,2.4.2.30 0003950 ic50=0.008uM -logKd/Ki=8.10, IC50=0.008uM IC50=8.0nM O95271 23316926 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPEH 4i9i B 2.4 BS02 1DY B 1 H1184 G1185 F1188 A1191 G1196 D1198 H1201 I1212 Y1213 F1214 A1215 S1221 Y1224 E1291 H81 G82 F85 A88 G93 D95 H98 I109 Y110 F111 A112 S118 Y121 E188 2.4.2.-,2.4.2.30 0003950 ic50=0.008uM IC50=8.0nM O95271 23316926 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPE 4i9i C 2.4 BS02 1DY C 1 H1184 G1185 F1188 I1192 G1196 D1198 H1201 I1212 Y1213 F1214 A1215 S1221 Y1224 E1291 H79 G80 F83 I87 G91 D93 H96 I107 Y108 F109 A110 S116 Y119 E186 2.4.2.-,2.4.2.30 0003950 ic50=0.008uM IC50=8.0nM O95271 23316926 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPE 4i9i D 2.4 BS02 1DY D 1 H1184 G1185 F1188 A1191 G1196 D1198 H1201 I1212 Y1213 F1214 A1215 K1220 S1221 Y1224 E1291 H80 G81 F84 A87 G92 D94 H97 I108 Y109 F110 A111 K116 S117 Y120 E183 2.4.2.-,2.4.2.30 0003950 ic50=0.008uM IC50=8.0nM O95271 23316926 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPLAYAEYVIYRGEQAYPEYLITYQIMKPE