4i4e A 1.55 BS01 1BQ A 1 R426 I428 A452 M499 E500 C502 L504 G505 L553 R13 I15 A38 M85 E86 C88 L90 G91 L139 D546 A548 R550 N551 D564 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.5uM -logKd/Ki=6.30, IC50=0.5uM Q05397 23414845 1000 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPNPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ