2hk5 A 2.0 BS01 1BM A 1 L251 A271 K273 E288 I314 T316 F318 M319 G322 A368 N369 L371 D382 L23 A43 K45 E60 I86 T88 F90 M91 G94 A140 N141 L143 D154 D364 R366 A368 N369 D382 F402 D136 R138 A140 N141 D154 F174 2.7.10.2 0004672,0004713,0005524,0006468 ic50=46nM -logKd/Ki=7.34, IC50=46nM IC50=46nM P08631 16997556 499 AQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDF