4i0t A 1.7 BS01 1B6 A 1 L377 A400 M448 M450 A451 P455 L501 S511 L15 A38 M80 M82 A83 P87 L133 S143 D494 A496 R498 N499 D512 D126 A128 R130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 ic50=26nM -logKd/Ki=7.59, IC50=26nM IC50=26nM P43405 23350847 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH