4hf4 A 2.0 BS02 15H A 1 Y514 I682 Y683 F686 P702 M703 E711 V712 G715 Q716 F719 Y73 I241 Y242 F245 P261 M262 E270 V271 G274 Q275 F278 3.1.4.17 0004114,0007165,0008081 ic50=2.4nM -logKd/Ki=8.62, Ki=2.4nM IC50=2.4nM Q9Y233 23149228 1012 TSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4hf4 B 2.0 BS02 15H B 1 Y514 I682 Y683 F686 P702 M703 E711 V712 G715 Q716 F719 Y63 I231 Y232 F235 P251 M252 E260 V261 G264 Q265 F268 3.1.4.17 0004114,0007165,0008081 ic50=2.4nM IC50=2.4nM Q9Y233 23149228 810 FTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE