4gih A 2.0 BS01 0X5 A 1 L903 G904 E905 V911 I960 Y980 V981 G984 L1030 L14 G15 E16 V22 I71 Y91 V92 G95 L141 N1023 A1025 R1027 N1028 D1041 E1050 P1064 N134 A136 R138 N139 D152 E161 P175 2.7.10.2 0004672,0005524,0006468 Ki=0.0048uM -logKd/Ki=8.32, Ki=0.0048uM Ki=4.8nM P29597 23867602 1201 TVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYR 4gmy A 2.403 BS01 0X5 A 1 V863 Y931 L932 P933 G935 L983 V31 Y99 L100 P101 G103 L151 D976 A978 R980 N981 D994 S1016 D144 A146 R148 N149 D162 S184 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.028uM -logKd/Ki=7.55, Ki=0.028uM Ki=28nM, EC50=1700nM O60674 23867602 1201 SGAFEDRDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG