3ika A 2.9 BS01 0UN A 1 L718 G719 V726 A743 M790 L792 M793 G796 C797 D800 L844 L23 G24 V31 A48 M95 L97 M98 G101 C102 D105 L149 D837 A839 R841 N842 D855 G874 D142 A144 R146 N147 D160 G179 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=7.85, IC50=14nM IC50=<1nM, Kd=1.2nM, EC50=68nM P00533 20033049 1797 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHEEDMDDVVDADEYLIPQ 5x2k A 3.201 BS01 0UN A 1 L718 M793 P794 G796 L844 L23 M96 P97 G99 L147 D837 A839 R841 N842 D855 D140 A142 R144 N145 D158 2.7.10.1 0004672,0004713,0005524,0006468 IC50=<1nM, Kd=1.2nM, EC50=68nM P00533 29568384 1101 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPDSNFYRALMDEEDMDDVVDADEYLIPQ 7zyn A 2.3 BS01 0UN A 1 L718 G719 F723 V726 A743 M790 M793 P794 G796 L844 L22 G23 F27 V30 A47 M90 M93 P94 G96 L144 2.7.10.1 0004672,0004713,0005524,0006468 P00533 37197473 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGSLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAAAAEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPDSNFYRALMDEEDMDDVVDADEYLI