4f1l A 1.9 BS01 0RY A 1 H1601 G1602 N1624 Y1633 F1634 A1635 Y1640 S1641 Y1646 H68 G69 N91 Y100 F101 A102 Y107 S108 Y113 2.4.2.- 0003950 -logKd/Ki=5.12, Kd=7.6uM IC50=>20000nM, Kd=7600nM Q460N5 22823910 1801 QNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGKNAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 4f1l B 1.9 BS01 0RY B 1 H1601 G1602 Y1633 F1634 A1635 S1641 Y1646 H70 G71 Y94 F95 A96 S102 Y107 2.4.2.- 0003950 IC50=>20000nM, Kd=7600nM Q460N5 22823910 1801 KQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 4f1l C 1.9 BS01 0RY C 1 H1601 G1602 N1624 V1626 Y1633 F1634 A1635 Y1640 S1641 Y1646 H68 G69 N91 V93 Y100 F101 A102 Y107 S108 Y113 2.4.2.- 0003950 IC50=>20000nM, Kd=7600nM Q460N5 22823910 1801 QNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGKNAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 4f1l C 1.9 BS02 0RY D 1 T1645 Y1646 T112 Y113 2.4.2.- 0003950 IC50=>20000nM, Kd=7600nM Q460N5 22823910 1801 QNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGKNAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 4f1l D 1.9 BS01 0RY D 1 H1601 G1602 V1626 Y1633 F1634 A1635 Y1640 S1641 Y1646 H68 G69 V91 Y98 F99 A100 Y105 S106 Y111 2.4.2.- 0003950 IC50=>20000nM, Kd=7600nM Q460N5 22823910 1801 QNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK