4ebw A 2.65 BS01 0PF A 1 L534 L537 H544 R550 N551 L562 G563 D604 M607 L122 L125 H132 R138 N139 L150 G151 D177 M180 D546 A548 R550 N551 D564 K583 D134 A136 R138 N139 D152 K156 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=5.06, IC50=8.7uM IC50=>30000nM Q05397 22819505 700 STRDYEIQRERIELGRCIGEGQFGDVHQGIYMSNPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLKLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ