1ca8 B 2.1 BS03 0KV B 1 H57 Y60A W60D I174 D189 C191 S195 S214 W215 G216 G219 H42 Y46 W49 I170 D190 C192 S196 S217 W218 G219 G221 H57 D102 E192 G193 D194 S195 G196 H42 D98 E193 G194 D195 S196 G197 3.4.21.5 0004252,0005509,0006508,0007596 -logKd/Ki=9.49, Ki=0.32nM IC50=0.67nM P00734 9724521 248 IVEGSDAEIGMSPWQVMLFRKPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1yyy 1 2.1 BS02 0KV 1 1 H57 D189 S190 C191 S195 S214 W215 G216 S217 G219 H40 D171 S172 C173 S177 S192 W193 G194 S195 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 -logKd/Ki=5.09, Ki=8100nM P00760 9724521 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN