4dfn A 2.48 BS01 0K1 A 1 L377 F382 V385 A400 M448 A451 P455 K458 L501 D512 L15 F20 V23 A38 M81 A84 P88 K91 L134 D145 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.02uM -logKd/Ki=7.70, IC50=0.02uM IC50=20nM P43405 22425453 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNE