4k4a A 1.89 BS01 0FQ A 1 Q48 P49 L53 H54 G55 H89 V90 R91 S92 Q48 P49 L53 H54 G55 H89 V90 R91 S92 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a A 1.89 BS02 0FQ C 1 S67 V81 G82 L136 S67 V81 G82 L136 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a A 1.89 BS03 0FQ D 1 H106 G108 S109 R110 H111 H106 G108 S109 R110 H111 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a B 1.89 BS01 0FQ A 1 S67 V81 G82 S67 V81 G82 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a B 1.89 BS02 0FQ B 1 H106 G108 S109 R110 H111 H106 G108 S109 R110 H111 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a B 1.89 BS03 0FQ C 1 Q48 P49 H54 G55 H89 V90 R91 S92 Q48 P49 H54 G55 H89 V90 R91 S92 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a C 1.89 BS01 0FQ B 1 Q48 P49 H54 G55 H89 V90 R91 S92 Q48 P49 H54 G55 H89 V90 R91 S92 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a C 1.89 BS02 0FQ C 1 H106 G108 S109 R110 H111 H106 G108 S109 R110 H111 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a C 1.89 BS03 0FQ D 1 S67 V81 G82 L136 S67 V81 G82 L136 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a D 1.89 BS01 0FQ A 1 H106 G108 S109 R110 H111 H106 G108 S109 R110 H111 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a D 1.89 BS02 0FQ B 1 E63 S67 V81 G82 L136 E63 S67 V81 G82 L136 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4a D 1.89 BS03 0FQ D 1 Q48 P49 H54 G55 H89 V90 R91 S92 Q48 P49 H54 G55 H89 V90 R91 S92 3.1.2.28 0005829,0009234,0016289,0016787,0016790,0061522 Ki=7.8uM P77781 25010423 201 MIWKRKITLEALNAMGEGNMVGFLDIRFEHIGDDTLEATMPVDSRTKQPFGLLHGGASVVLAESIGSVAGYLCTEGEQKVVGLEINANHVRSAREGRVRGVCKPLHLGSRHQVWQIEIFDEKGRLCCSSRLTTAIL 4k4c A 1.85 BS01 0FQ A 1 Q48 P49 F50 H54 G55 H89 H90 R91 P92 Q48 P49 F50 H54 G55 H89 H90 R91 P92 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c A 1.85 BS02 0FQ B 1 H106 G108 R109 Q110 N111 H106 G108 R109 Q110 N111 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c A 1.85 BS03 0FQ D 1 E63 S67 M68 V81 G82 E63 S67 M68 V81 G82 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c B 1.85 BS01 0FQ A 1 G108 R109 Q110 N111 G108 R109 Q110 N111 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c B 1.85 BS02 0FQ B 1 Q48 P49 F50 L53 H54 G55 H89 H90 R91 P92 Q48 P49 F50 L53 H54 G55 H89 H90 R91 P92 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c B 1.85 BS03 0FQ C 1 S67 M68 V81 G82 S67 M68 V81 G82 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c C 1.85 BS01 0FQ B 1 S67 M68 V81 G82 L136 S67 M68 V81 G82 L136 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c C 1.85 BS02 0FQ C 1 Q48 P49 L53 H54 G55 H89 H90 R91 P92 Q48 P49 L53 H54 G55 H89 H90 R91 P92 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c C 1.85 BS03 0FQ D 1 G108 R109 Q110 G108 R109 Q110 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c D 1.85 BS01 0FQ A 1 S67 M68 V81 G82 S67 M68 V81 G82 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c D 1.85 BS02 0FQ C 1 G108 R109 Q110 N111 G108 R109 Q110 N111 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4k4c D 1.85 BS03 0FQ D 1 Q48 P49 L53 H54 G55 H89 H90 R91 P92 Q48 P49 L53 H54 G55 H89 H90 R91 P92 3.1.2.- 0005515,0005737,0005829,0009239,0016289,0016787,0016788,0016790,0042802,0061522 Ki=65uM P0A8Y8 25010423 201 MIWKRHLTLDELNATSDNTMVAHLGIVYTRLGDDVLEAEMPVDTRTHQPFGLLHGGASAALAETLGSMAGFMMTRDGQCVVGTELNATHHRPVSEGKVRGVCQPLHLGRQNQSWEIVVFDEQGRRCCTCRLGTAVLG 4qd8 C 1.616 BS01 0FQ C 1 H108 G110 R111 T112 T113 H107 G109 R110 T111 T112 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 201 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 C 1.616 BS02 0FQ C 2 Q49 P50 H55 H91 L92 R93 R96 Q48 P49 H54 H90 L91 R92 R95 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 202 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 C 1.616 BS03 0FQ D 2 E64 S68 V83 G84 E63 S67 V82 G83 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 202 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 D 1.616 BS01 0FQ C 2 E64 S68 V83 G84 E63 S67 V82 G83 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 202 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 D 1.616 BS02 0FQ D 1 H108 G110 R111 T112 T113 H107 G109 R110 T111 T112 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 201 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 D 1.616 BS03 0FQ D 2 Q49 P50 H55 G56 H91 L92 R93 G94 Q48 P49 H54 G55 H90 L91 R92 G93 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 202 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 E 1.616 BS01 0FQ C 1 Q49 P50 H55 G56 H91 L92 R93 K126 Q48 P49 H54 G55 H90 L91 R92 K125 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 201 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 E 1.616 BS02 0FQ C 2 H108 G110 R111 T112 T113 H107 G109 R110 T111 T112 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 202 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 E 1.616 BS03 0FQ D 1 S68 G84 S67 G83 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 201 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 F 1.616 BS01 0FQ C 1 E64 S68 M69 V83 G84 E63 S67 M68 V82 G83 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 201 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 F 1.616 BS02 0FQ D 1 Q49 P50 H55 G56 H91 L92 R93 Q48 P49 H54 G55 H90 L91 R92 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 201 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL 4qd8 F 1.616 BS03 0FQ D 2 H108 G110 R111 T112 T113 H107 G109 R110 T111 T112 3.1.2.- 0005829,0016289,0016787,0061522 Q9I3A4 202 SLWRQTPDLEQLNASQKNSIGDLLGIRFEAFDDESLTASMPVDSRTHQPFGLLHGGASVVLAESLGSMASYLCVDTSQYYCVGLEVNANHLRGLRSGRVTAVARAIHLGRTTHVWDIRLSGDDGKPSCIARLTMAVVPL