3up7 A 3.05 BS01 0C9 A 1 R137 L139 G140 V147 A160 A213 G216 R220 D274 R14 L16 G17 V24 A37 A90 G93 R97 D151 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=8.21, IC50=6.1nM IC50=6.1nM, Kd=34nM O14965 22803810 1 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANS