3uoh A 2.8002 BS01 0C4 A 1 R137 L139 L194 Y212 A213 G216 T217 R220 L263 V279 R12 L14 L69 Y87 A88 G91 T92 R95 L138 V154 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T167 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=7.89, Kd=13nM IC50=2.1nM, Kd=13nM O14965 22248356 2 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3uoh B 2.8002 BS01 0C4 B 1 L194 Y212 A213 G216 T217 R220 L263 V279 L69 Y87 A88 G91 T92 R95 L138 V154 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T167 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 IC50=2.1nM, Kd=13nM O14965 22248356 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK