3tzm A 1.7 BS01 085 A 1 G214 A230 K232 L278 S280 Y282 H283 K337 L340 D351 G15 A31 K33 L79 S81 Y83 H84 K138 L141 D152 D333 K335 N338 D351 T375 D134 K136 N139 D152 T174 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 -logKd/Ki=7.77, Ki=17nM IC50=94nM, Ki=17nM, EC50=172nM P36897 21983015 1 TIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLS