3dct A 2.5 BS02 064 A 1 M265 F284 L287 T288 M290 H294 M328 F329 R331 I335 H447 W454 W469 M22 F41 L44 T45 M47 H51 M85 F86 R88 I92 H204 W211 W226 ? 0004879,0032052,0038183 -logKd/Ki=6.95, IC50=0.112uM EC50=65nM, IC50=20nM Q96RI1 18621523 1 ELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEEFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEERIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 6a60 A 3.05 BS02 064 A 1 Q263 M290 H294 M328 F329 R331 I335 M365 Y369 H447 W454 F461 Q20 M42 H46 M80 F81 R83 I87 M113 Y117 H195 W202 F209 ? 0003677,0004879,0006355,0032052,0038183 EC50=65nM, IC50=20nM Q96RI1 30275017 501 ELTPDQQTLLHFIMDSYNKQRMPQEITNKFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLSDLLEERIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFAELLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLEEIWDV