1ztq A 2.0 BS06 033 A 1 L159 L160 A161 H197 E198 H201 H207 G212 L214 F216 P217 I218 Y219 T220 F227 P230 L78 L79 A80 H116 E117 H120 H126 G131 L133 F135 P136 I137 Y138 T139 F146 P149 H197 E198 H201 H207 H116 E117 H120 H126 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=1.3nM -logKd/Ki=8.89, IC50=1.3nM IC50=1.3nM P45452 16005220 601 YNVFLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGP 1ztq B 2.0 BS06 033 B 1 L159 L160 A161 H197 E198 H207 L214 F216 P217 I218 Y219 T220 L76 L77 A78 H114 E115 H124 L131 F133 P134 I135 Y136 T137 H197 E198 H201 H207 H114 E115 H118 H124 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=1.3nM IC50=1.3nM P45452 16005220 602 YNVKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGP 1ztq C 2.0 BS06 033 C 1 L159 L160 A161 L193 H197 E198 H207 G212 L214 F216 P217 I218 Y219 P230 L78 L79 A80 L112 H116 E117 H126 G131 L133 F135 P136 I137 Y138 P140 H197 E198 H201 H207 H116 E117 H120 H126 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=1.3nM IC50=1.3nM P45452 16005220 603 YNVFLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTPDDDVQGIQSLYGP 1ztq D 2.0 BS06 033 D 1 L159 L160 A161 V194 H197 E198 H207 G212 L214 F216 P217 I218 Y219 F227 L78 L79 A80 V113 H116 E117 H126 G131 L133 F135 P136 I137 Y138 F140 H197 E198 H201 H207 H116 E117 H120 H126 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=1.3nM IC50=1.3nM P45452 16005220 604 YNVFLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTFMLPDDDVQGIQSLYGP