3g90 X 2.4 BS01 J72 X 1 I70 V78 E147 M149 D150 A151 N152 V196 L206 I25 V31 E100 M102 D103 A104 N105 V149 L159 N194 D207 N147 D160 2.7.11.24 0004672,0004707,0005524,0006468 Ki=0.44uM -logKd/Ki=6.36, Ki=0.44uM P53779 19361991 1 NQFYSVEVGDSTFTVLKRYQNLKPIGSQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQIQLDEREHTIEEWKELIYKEVMN