1y0x X 3.1 BS01 T44 X 1 F272 I276 A279 R282 M310 M313 R316 L346 H435 M442 F455 F459 F62 I66 A69 R72 M100 M103 R106 L136 H225 M232 F245 F249 ? 0003677,0004879,0006355 -logKd/Ki=8.70, Kd=2nM EC50=240nM P10828 15466465 500 SHMEELQKSIGHKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFE