3h4v F 2.4 BS01 NAP F 1 R17 L18 H36 Y37 H38 R39 S40 L66 N109 A110 S111 S112 M179 V180 D181 K198 P224 L226 S227 R13 L14 H32 Y33 H34 R35 S36 L62 N99 A100 S101 S102 M161 V162 D163 K180 P206 L208 S209 R17 D181 Y194 R13 D163 Y176 1.5.1.33 0004155,0005829,0006729,0016491,0031427,0047040 Q01782 18245389 300 TVPVALVTGAAKRLGRSIAEGLHAEGYAVCLHYHRSAAEANALSATLNARRPNSAITVQADLSNVATAPSAPVTLFTRCAELVAACYTHWGRCDVLVNNASSFYPTPLLRNDGDREAMETATADLFGSNAIAPYFLIKAFAHRVAGTPAKHRGTNYSIINMVDAMTNQPLLGYTIYTMAKGALEGLTRSAALELAPLQIRVNGVGPGLSVLVDDMPPAVWEGHRSKVPLYQRDSSAAEVSDVVIFLCSSKAKYITGTCVKVDGGYSLTRA 3h4v F 2.4 BS02 DVP F 1 S111 F113 L188 Y191 Y194 S101 F103 L170 Y173 Y176 R17 D181 Y194 R13 D163 Y176 1.5.1.33 0004155,0005829,0006729,0016491,0031427,0047040 Ki=0.1uM Ki=100nM Q01782 18245389 301 TVPVALVTGAAKRLGRSIAEGLHAEGYAVCLHYHRSAAEANALSATLNARRPNSAITVQADLSNVATAPSAPVTLFTRCAELVAACYTHWGRCDVLVNNASSFYPTPLLRNDGDREAMETATADLFGSNAIAPYFLIKAFAHRVAGTPAKHRGTNYSIINMVDAMTNQPLLGYTIYTMAKGALEGLTRSAALELAPLQIRVNGVGPGLSVLVDDMPPAVWEGHRSKVPLYQRDSSAAEVSDVVIFLCSSKAKYITGTCVKVDGGYSLTRA