2gpv F 2.85 BS01 OHT F 1 C269 A272 D273 E275 M306 Y326 F435 C37 A40 D41 E43 M74 Y94 F203 ? IC50=1350nM, EC50=15nM P62508 16990259 505 PYNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKL