7jxp E 2.16 BS01 JBJ E 1 V726 A743 I744 K745 I759 R776 L777 L788 M790 D855 F856 L858 V27 A44 I45 K46 I60 R77 L78 L89 M91 D156 F157 L159 2.7.10.1 0004672,0004713,0005524,0006468 IC50=>1000nM P00533 1101 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDPSPTDSNFYRALMDEEDM 7jxp E 2.16 BS02 YY3 E 1 L718 V726 L792 M793 G796 C797 D800 L844 D855 L19 V27 L93 M94 G97 C98 D101 L145 D156 2.7.10.1 0004672,0004713,0005524,0006468 IC50=2.0nM, Ki=14nM, EC50=6.0nM P00533 1102 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDPSPTDSNFYRALMDEEDM