4e4l E 2.0 BS01 0NH A 2 L881 G882 E883 V889 A906 M956 F958 L959 R1007 N1008 L1010 D1021 L18 G19 E20 V26 A43 M84 F86 L87 R135 N136 L138 D149 N1008 D1021 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 EC50=210nM, Ki=1.7nM P23458 22591402 1202 EVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK