1ere E 3.1 BS01 EST E 1 E353 F404 H524 L525 E43 F94 H211 L212 ? IC50=1.3nM, Kd=0.2nM, EC50=0.75nM, Ki=0.21nM P03372 9338790 600 SLALSLTADQMVSALLDAEPPILYSEFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHR