4r6e D 2.2 BS01 3JD D 1 D766 H862 G863 G888 Y889 Y896 F897 A898 S904 Y907 D104 H200 G201 G226 Y227 Y234 F235 A236 S242 Y245 S904 Y907 E988 S242 Y245 E326 2.4.2.-,2.4.2.30 0003950 ic50=132nM IC50=132nM, Ki=3.2nM, EC50=31000nM P09874 28001384 1101 SKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK