3bzu D 2.25 BS01 NAP D 1 G41 S43 K44 G45 I46 R66 T92 M93 N119 I121 V168 S170 Y183 K187 L215 L217 I218 T220 T222 A223 G16 S18 K19 G20 I21 R41 T65 M66 N92 I94 V141 S143 Y156 K160 L188 L190 I191 T193 T195 A196 S170 Y183 K187 S143 Y156 K160 1.1.1.146,1.1.1.201 0005496,0005783,0005789,0006706,0008202,0016020,0016491,0030324,0042803,0043231,0047022,0050661,0070524,0102196 P28845 18069989 4 EFRPEMLQGKKVIVTGASKGIGREMAYHLAKMGAHVVVTARETLQKVVSHCLELGAASAHYIAGTMEDMTFAEQFVAQAGKLMGGLDMLILNHITNTSLNLFHDDIHHVRKSMEVNFLSYVVLTVAALPMLKQSNGSIVVVSSLAGKVAYPMVAAYSASKFALDGFFSSIRKEYSVSRVNVSITLCVLGLIDTETAMKAVSGIVHMQAAPKEECALEIIKGGALRQEEVYYDSSLWTTLLIRNPSRKILEFLYS 3bzu D 2.25 BS02 A21 D 1 T124 L171 A172 Y183 L217 M233 T97 L144 A145 Y156 L190 M206 S170 Y183 K187 S143 Y156 K160 1.1.1.146,1.1.1.201 0005496,0005783,0005789,0006706,0008202,0016020,0016491,0030324,0042803,0043231,0047022,0050661,0070524,0102196 ic50=14nM Ki=22nM P28845 18069989 293 EFRPEMLQGKKVIVTGASKGIGREMAYHLAKMGAHVVVTARETLQKVVSHCLELGAASAHYIAGTMEDMTFAEQFVAQAGKLMGGLDMLILNHITNTSLNLFHDDIHHVRKSMEVNFLSYVVLTVAALPMLKQSNGSIVVVSSLAGKVAYPMVAAYSASKFALDGFFSSIRKEYSVSRVNVSITLCVLGLIDTETAMKAVSGIVHMQAAPKEECALEIIKGGALRQEEVYYDSSLWTTLLIRNPSRKILEFLYS