2cht D 2.2 BS01 TSA D 1 R7 E78 R90 Y108 R6 E77 R89 Y107 R7 R63 C75 E78 R90 Y108 R6 R62 C74 E77 R89 Y107 5.4.99.5 0004106,0005737,0008652,0009073,0016853,0046417 Ki=3uM P19080 8378335 206 MIRGIRGATTVERDTEEEILQKTKQLLEKIIEENHTKPEDVVQMLLSATPDLHAVFPAKAVRELSGWQYVPVTCMQEMDVTGGLKKCIRVMMTVQTDVPQDQIRHVYLEKAVVL 2cht D 2.2 BS02 TSA E 1 F57 A59 R63 T74 C75 F56 A58 R62 T73 C74 R7 R63 C75 E78 R90 Y108 R6 R62 C74 E77 R89 Y107 5.4.99.5 0004106,0005737,0008652,0009073,0016853,0046417 Ki=3uM P19080 8378335 204 MIRGIRGATTVERDTEEEILQKTKQLLEKIIEENHTKPEDVVQMLLSATPDLHAVFPAKAVRELSGWQYVPVTCMQEMDVTGGLKKCIRVMMTVQTDVPQDQIRHVYLEKAVVL 2cht F 2.2 BS01 TSA D 1 F57 A59 K60 C75 F56 A58 K59 C74 R7 R63 C75 E78 R90 Y108 R116 R6 R62 C74 E77 R89 Y107 R115 5.4.99.5 0004106,0005737,0008652,0009073,0016853,0046417 Ki=3uM P19080 8378335 206 MIRGIRGATTVERDTEEEILQKTKQLLEKIIEENHTKPEDVVQMLLSATPDLHAVFPAKAVRELSGWQYVPVTCMQEMDVTGGLKKCIRVMMTVQTDVPQDQIRHVYLEKAVVLRPDL