1o5w D 3.2 BS01 FAD D 1 I3019 G3022 S3024 E3043 A3044 R3045 G3050 R3051 G3066 G3067 A3068 Y3069 P3243 V3244 I3273 K3305 W3397 Y3402 C3406 Y3407 G3434 T3435 G3443 Y3444 M3445 A3448 I10 G13 S15 E34 A35 R36 G41 R42 G57 G58 A59 Y60 P234 V235 I264 K296 W388 Y393 C397 Y398 G425 T426 G434 Y435 M436 A439 G3071 R3206 K3305 G62 R197 K296 1.4.3.21,1.4.3.4 0005739,0005741,0006584,0008131,0009967,0016491,0042420,0042424,0042428,0042443,0050660,0051378,0052595,0097621 P21396 15050826 3652 AGHMFDVVVIGGGISGLAAAKLLSEYKINVLVLEARDRVGGRTYTVRNEHVKWVDVGGAYVGPTQNRILRLSKELGIETYKVNVNERLVQYVKGKTYPFRGAFPPVWNPLAYLDYNNLWRTMDEMGKEIPVDAPWQARHAQEWDKMTMKDLIDKICWTKTAREFAYLFVNINVTSEPHEVSALWFLWYVRQCGGTARIFSVTNGGQERKFVGGSGQVSEQIMGLLGDKVKLSSPVTYIDQTDDNIIVETLNHEHYECKYVISAIPPILTAKIHFKPELPPERNQLIQRLPMGAVIKCMVYYKEAFWKKKDYCGCMIIEDEEAPIAITLDDTKPDGSLPAIMGFILARKADRLAKLHKDIRKRKICELYAKVLGSQEALYPVHYEEKNWCEEQYSGGCYTAYFPPGIMTQYGRVIRQPVGRIYFAGTETATQWSGYMEGAVEAGERAAREVLNALGKVAKKDIWVEEPESKDVPAIEITHTFLERNLPSVPGLLKITGVSTSVALLC 1o5w D 3.2 BS02 MLG D 1 I3180 F3208 Q3215 C3323 I3335 T3336 Y3407 Y3444 I171 F199 Q206 C314 I326 T327 Y398 Y435 G3071 R3206 K3305 G62 R197 K296 1.4.3.21,1.4.3.4 0005739,0005741,0006584,0008131,0009967,0016491,0042420,0042424,0042428,0042443,0050660,0051378,0052595,0097621 IC50=2050nM, Ki=1200nM P21396 15050826 3709 AGHMFDVVVIGGGISGLAAAKLLSEYKINVLVLEARDRVGGRTYTVRNEHVKWVDVGGAYVGPTQNRILRLSKELGIETYKVNVNERLVQYVKGKTYPFRGAFPPVWNPLAYLDYNNLWRTMDEMGKEIPVDAPWQARHAQEWDKMTMKDLIDKICWTKTAREFAYLFVNINVTSEPHEVSALWFLWYVRQCGGTARIFSVTNGGQERKFVGGSGQVSEQIMGLLGDKVKLSSPVTYIDQTDDNIIVETLNHEHYECKYVISAIPPILTAKIHFKPELPPERNQLIQRLPMGAVIKCMVYYKEAFWKKKDYCGCMIIEDEEAPIAITLDDTKPDGSLPAIMGFILARKADRLAKLHKDIRKRKICELYAKVLGSQEALYPVHYEEKNWCEEQYSGGCYTAYFPPGIMTQYGRVIRQPVGRIYFAGTETATQWSGYMEGAVEAGERAAREVLNALGKVAKKDIWVEEPESKDVPAIEITHTFLERNLPSVPGLLKITGVSTSVALLC