1mx1 D 2.4 BS01 SIA D 1 G4052 K4078 N4079 P4085 Y4118 G31 K57 N58 P64 Y97 G4142 G4143 S4221 A4222 E4354 H4468 G121 G122 S200 A201 E333 H446 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 P23141 12725862 482 SPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK 1mx1 D 2.4 BS02 THA D 1 S4221 L4304 L4363 H4468 S200 L283 L341 H446 G4142 G4143 S4221 A4222 E4354 H4468 G121 G122 S200 A201 E333 H446 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 IC50=>100000nM, Ki=>100000nM P23141 12725862 4 SPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK