4rxd C 2.0 BS01 RIS C 1 D103 R112 Q172 K212 T213 D255 K269 D93 R102 Q162 K202 T203 D245 K259 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=300nM -logKd/Ki=6.52, IC50=300nM Q86C09 25815158 1600 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 4rxd C 2.0 BS02 MG C 1 D103 D107 D93 D97 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Q86C09 25815158 1601 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 4rxd C 2.0 BS03 MG C 2 D103 D107 D93 D97 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Q86C09 25815158 1603 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK