3cm2 C 2.5 BS01 ZN C 1 C300 C303 H320 C327 C48 C51 H68 C75 2.3.2.27 P98170 18851976 502 STNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 3cm2 C 2.5 BS02 X23 C 1 L292 K297 V298 G306 L307 T308 D309 W310 E314 W323 L40 K45 V46 G54 L55 T56 D57 W58 E62 W71 2.3.2.27 Ki=340nM IC50=110nM P98170 18851976 600 STNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 3cm2 C 2.5 BS03 X23 F 1 H346 E349 H94 E97 2.3.2.27 Ki=340nM IC50=110nM P98170 18851976 600 STNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 3cm2 G 2.5 BS01 X23 C 1 H346 E349 H93 E96 2.3.2.27 Ki=340nM IC50=110nM P98170 18851976 600 TNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVRT