2hyy C 2.4 BS01 STI C 1 Y253 A269 K271 E286 M290 V299 I313 T315 F317 M318 I360 H361 L370 A380 D381 F382 Y21 A37 K39 E53 M57 V66 I80 T82 F84 M85 I127 H128 L137 A147 D148 F149 D363 A365 R367 N368 D381 P402 D130 A132 R134 N135 D148 P166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=170nM IC50=38nM, Kd=44nM, Ki=13nM, EC50=7e+1nM P00519 17164530 600 DKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKETMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQ