2cht B 2.2 BS02 TSA C 1 F57 A59 V73 T74 C75 F56 A58 V72 T73 C74 R7 R63 C75 E78 R90 Y108 R116 R6 R62 C74 E77 R89 Y107 R115 5.4.99.5 0004106,0005737,0008652,0009073,0016853,0046417 Ki=3uM P19080 8378335 202 MIRGIRGATTVERDTEEEILQKTKQLLEKIIEENHTKPEDVVQMLLSATPDLHAVFPAKAVRELSGWQYVPVTCMQEMDVTGGLKKCIRVMMTVQTDVPQDQIRHVYLEKAVVLRPD 2cht C 2.2 BS01 TSA A 1 F57 A59 K60 R63 T74 C75 F56 A58 K59 R62 T73 C74 R7 R63 C75 E78 R90 Y108 R116 R6 R62 C74 E77 R89 Y107 R115 5.4.99.5 0004106,0005737,0008652,0009073,0016853,0046417 Ki=3uM P19080 8378335 203 MIRGIRGATTVERDTEEEILQKTKQLLEKIIEENHTKPEDVVQMLLSATPDLHAVFPAKAVRELSGWQYVPVTCMQEMDVTGGLKKCIRVMMTVQTDVPQDQIRHVYLEKAVVLRPDL 2cht C 2.2 BS02 TSA C 1 R7 E78 R90 Y108 L115 R6 E77 R89 Y107 L114 R7 R63 C75 E78 R90 Y108 R116 R6 R62 C74 E77 R89 Y107 R115 5.4.99.5 0004106,0005737,0008652,0009073,0016853,0046417 Ki=3uM P19080 8378335 202 MIRGIRGATTVERDTEEEILQKTKQLLEKIIEENHTKPEDVVQMLLSATPDLHAVFPAKAVRELSGWQYVPVTCMQEMDVTGGLKKCIRVMMTVQTDVPQDQIRHVYLEKAVVLRPDL