7jxm B 2.192 BS01 YY3 B 1 L718 G719 V726 A743 M793 G796 C797 D800 L18 G19 V26 A43 M93 G96 C97 D100 2.7.10.1 0004672,0004713,0005524,0006468 IC50=2.0nM, Ki=14nM, EC50=6.0nM P00533 1101 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVD 7jxm B 2.192 BS02 9LL B 1 V726 A743 K745 I759 C775 R776 L777 L788 M790 D855 F856 L858 V26 A43 K45 I59 C75 R76 L77 L88 M90 D155 F156 L158 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 1102 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVD