6t8x B 2.81 BS01 B97 B 1 L70 L72 V78 K93 M138 C140 L141 D142 L193 T206 D207 L26 L28 V34 K49 M94 C96 L97 D98 L149 T162 D163 D186 K188 N191 D207 T226 D142 K144 N147 D163 T173 2.7.11.1 0004672,0005524,0006468 IC50=201nM, Ki=5.0nM P49137 401 QFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNHGLAISPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQST 6t8x B 2.81 BS02 MW8 B 1 F147 G259 Y260 P261 Y264 S265 N266 G268 F103 G206 Y207 P208 Y211 S212 N213 G215 D186 K188 N191 D207 T226 D142 K144 N147 D163 T173 2.7.11.1 0004672,0005524,0006468 P49137 403 QFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNHGLAISPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQST