6p1d B 2.4 BS01 ANP B 1 G719 S720 G721 V726 A743 K745 M790 M793 C797 D837 R841 N842 L844 D855 G18 S19 G20 V25 A42 K44 M89 M92 C96 D136 R140 N141 L143 D154 D837 R841 N842 D855 D136 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 P00533 31749909 1101 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDA 6p1d B 2.4 BS02 NQ1 B 1 A743 K745 M766 C775 R776 L788 M790 D855 F856 L858 L861 A42 K44 M65 C74 R75 L87 M89 D154 F155 L157 L160 D837 R841 N842 D855 D136 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=7.41, IC50=39nM IC50=>10000nM P00533 31749909 1102 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDA 6p1d B 2.4 BS03 MG B 1 N842 D855 N141 D154 D837 R841 N842 D855 D136 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 P00533 31749909 1103 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDA