6cjf B 1.63 BS01 FMN B 1 A96 G97 K100 S120 N145 N181 N212 K255 N284 T285 S305 G306 V333 G334 G335 Y356 T357 A54 G55 K58 S78 N103 N139 N170 K205 N234 T235 S255 G256 V283 G284 G285 Y306 T307 N145 F149 S215 K255 N284 N103 F107 S173 K205 N234 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 Q02127 29727569 501 RFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRRLEA 6cjf B 1.63 BS02 F54 B 1 Y38 M43 Q47 P52 A55 H56 A59 R136 Y356 T360 P364 Y3 M8 Q12 P17 A20 H21 A24 R94 Y306 T310 P314 N145 F149 S215 K255 N284 N103 F107 S173 K205 N234 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 ic50=0.0262uM IC50=26nM Q02127 29727569 503 RFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRRLEA 6cjf B 1.63 BS03 ZWI B 1 L58 F62 L23 F27 N145 F149 S215 K255 N284 N103 F107 S173 K205 N234 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 Q02127 29727569 504 RFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRRLEA 6cjf B 1.63 BS04 ZWI B 2 L84 R241 L42 R191 N145 F149 S215 K255 N284 N103 F107 S173 K205 N234 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 Q02127 29727569 505 RFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRRLEA