5uis B 2.5 BS01 8C1 B 1 E194 V200 A211 Y262 Y264 M265 G268 A315 L318 E30 V36 A47 Y88 Y90 M91 G94 A141 L144 D311 K313 A315 N316 D329 T351 D137 K139 A141 N142 D155 T170 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=146nM IC50=146nM Q9NWZ3 28498658 801 FHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAEELKQQFDQEIKVMAKCQHENLVELLGFSSDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT