4tw9 B 2.4 BS01 386 B 1 I23 A36 Y56 M82 L85 G86 P87 D91 L135 L293 I23 A36 Y56 M82 L85 G86 P87 D91 L135 L287 D128 K130 D128 K130 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.02uM -logKd/Ki=7.70, IC50=0.02uM P48730 25191940 1007 MELRVGNRYRLGNKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKF