4puz	B	2.085	BS01	CG9	B	1	L377 F382 V385 A400 M450 A451 E452 G454 P455 L501	L15 F20 V23 A38 M83 A84 E85 G87 P88 L134	D494 A496 R498 N499 D512 K533	D127 A129 R131 N132 D145 K163	2.7.10.2	0004672,0004713,0005524,0006468		ic50=7.7nM		IC50=377nM, EC50=125nM	P43405	24779514	701 	VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN