4ppa B 2.67 BS01 2VU A 1 I369 V377 I14 V22 D482 A484 R486 N487 D500 P521 D120 A122 R124 N125 D138 P141 2.7.10.2 0004672,0004713,0004715,0005524,0006468 IC50=210nM, Ki=1.1nM Q08881 24767842 701 SVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4ppa B 2.67 BS02 2VU B 1 A389 K391 F435 E436 F437 M438 E439 G441 L489 D500 A34 K36 F73 E74 F75 M76 E77 G79 L127 D138 D482 A484 R486 N487 D500 P521 D120 A122 R124 N125 D138 P141 2.7.10.2 0004672,0004713,0004715,0005524,0006468 IC50=210nM, Ki=1.1nM Q08881 24767842 701 SVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG