4mxo B 2.105 BS01 DB8 B 1 L273 A293 I294 K295 E310 V323 I336 T338 Y340 M341 S342 L393 L16 A36 I37 K38 E53 V66 I79 T81 Y83 M84 S85 L136 D386 R388 A390 N391 D404 F424 D129 R131 A133 N134 D147 F155 2.7.10.2 0004672,0004713,0005524,0006468 Kd=0.73nM IC50=3.8nM, Kd=1nM P12931 24292070 601 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGETGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKEPEERPTFEYLQAFLEDYFTSTEPQYQPGENL